专题：Phenothiazines and Benzothiazines Synthesis and Activities

This cluster of papers focuses on the biological activities, synthesis, and potential applications of phenothiazines and related compounds. It covers a wide range of topics including antimicrobial, anticancer, and neuroprotective properties, as well as the use of non-antibiotic drugs and the Smiles rearrangement in their synthesis. The cluster also explores the inhibition of DNA synthesis, antioxidant activity, and the potential role of phenothiazines in managing antibiotic-resistant infections.
最新文献
Advances in radical Smiles rearrangement

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Comparison Between Moxifloxacin and Chloramphenicol for the Treatment of Bacterial Eye Infections

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Synthesis of sildenafil and its derivatives bearing pyrazolo‐pyrimidinones scaffold

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Multi-component Crystal Strategy for Improving Water Solubility and Antifungal Activity of Climbazole

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Development and validation of a stability indicating UPLC-DAD method coupled with MS-TQD for ramipril and thymoquinone in bioactive SNEDDS with in silico toxicity analysis of ramipril degradation products

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Immobilization of Ni nanoparticles on pyridine-functionalized MWCNTs for indirect synthesis of benzimidazoles and quinazolinones, and their molecular docking studies as effective inhibitors of α-glucosidase

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Assessment of the Efficacy of the Antihistamine Drug Rupatadine Used Alone or in Combination against Mycobacteria

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Synthesis of Indolo[2,3/3,2-c]quinoline through Complementary PIDA/BF3·OEt2 as Well as Pd(0)-Mediated Intramolecular Cyclization of Isomeric N-((Aryl)-N-(phenylsulfonyl)indolyl)methylbenzenesulfonamides

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Synthesis, antimicrobial activity, and biofilm inhibition studies of 1,2,3-triazole-containing 2,3-dihydrothiazole

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Synthesis, Structural Properties and Biological Activities of Novel Hydrazones of 2-, 3-, 4-Iodobenzoic Acid

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近5年高被引文献
Antibiotic resistance: The challenges and some emerging strategies for tackling a global menace

review Full Text OpenAlex 770 FWCI80.37505221

Sulfonamide drugs: structure, antibacterial property, toxicity, and biophysical interactions

review Full Text OpenAlex 445 FWCI29.45479303

Liquid‐Assisted Grinding Mechanochemistry in the Synthesis of Pharmaceuticals

article Full Text OpenAlex 313 FWCI21.9917467

Late-stage diversification of indole skeletons through nitrogen atom insertion

article Full Text OpenAlex 309 FWCI53.13188985

Improved Solubility and Dissolution Rate of Ketoprofen by the Formation of Multicomponent Crystals with Tromethamine

article Full Text OpenAlex 254 FWCI31.24239497

Exploring Phytochemicals for Combating Antibiotic Resistance in Microbial Pathogens

review Full Text OpenAlex 231 FWCI29.08543389

Role of bacterial efflux pumps in antibiotic resistance, virulence, and strategies to discover novel efflux pump inhibitors

review Full Text OpenAlex 205 FWCI35.18721531

Drug repurposing for next-generation combination therapies against multidrug-resistant bacteria

review Full Text OpenAlex 189 FWCI11.60293974

The Development of Third-Generation Tetracycline Antibiotics and New Perspectives

review Full Text OpenAlex 165 FWCI29.07912975

Design and synthesis of hybrid compounds as novel drugs and medicines

review Full Text OpenAlex 152 FWCI18.70651201